PDB | 6xrp Crystal structure of GlpG in complex with peptide ketoamide inhibitor, Ac-RVWHA-ketoamide-phenylbutyl

Crystal structure of GlpG in complex with peptide ketoamide inhibitor, Ac-RVWHA-ketoamide-phenylbutyl

label Keywords
glpg, rhomboid protease, hydrolase-hydrolase inhibitor complex, membrane protein
event_note Published
12/25/2024
blur_on Resolution
2.4 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
N-(4-phenylbutyl)formamide

Original publication

import_contacts Title
Designed Parasite-Selective Rhomboid Inhibitors Block Invasion and Clear Blood-Stage Malaria.
import_contacts Journal
Cell Chem Biol 2020
import_contacts DOI
10.1016/j.chembiol.2020.08.011
person Authors
Baker, R.P., Gandhi, S., Stanchev, S., Strisovsky, K., Cho, S., Urban, S.

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