PDB | 8u3c TRPV1 in nanodisc

TRPV1 in nanodisc bound with PI-Br4 bound in Conformation 2 (monomer)

label Keywords
trpv1 in nanodisc bound with pi-br4 bound in conformation 2 (monomer), membrane protein
event_note Published
10/02/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
(2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION

Original publication

import_contacts Title
Structural basis of TRPV1 modulation by endogenous bioactive lipids.
import_contacts Journal
Nat.Struct.Mol.Biol. 2024
import_contacts DOI
10.1038/s41594-024-01299-2
person Authors
Frost, A., Mancino, A., Moss 3rd, F.R., Cheng, Y., Julius, D., Arnold, W.R.

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