PDB | 8jwz Crystal structure of A2AR-T4L in complex with AB928
Crystal structure of A2AR-T4L in complex with AB928
label Keywords
adenosine receptor, inhibitor, complex, signaling protein
event_note Published
10/23/2024
blur_on Resolution
2.37 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
OLEIC ACID, SODIUM ION, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3-[2-azanyl-6-[1-[[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]methyl]-1,2,3-triazol-4-yl]pyrimidin-4-yl]-2-methyl-benzenecarbonitrile, DI(HYDROXYETHYL)ETHER, CHOLESTEROL
Original publication
import_contacts Title
Structural insight into the dual-antagonistic mechanism of AB928 on adenosine A 2 receptors.
import_contacts Journal
Sci China Life Sci 2024
import_contacts DOI
10.1007/s11427-023-2459-8
person Authors
Chen, Y., Zhang, Q., Weng, Y., Liu, M., Yang, H., Zhu, C., Lu, W., Xie, Q., Xu, Y., Song, G., Wang, Y., Yang, X.
Member of
copyrightData provided by Research Collaboration for Structural Biology, Chen, Y., Zhang, Q., Weng, Y., Liu, M., Yang, H., Zhu, C., Lu, W., Xie, Q., Xu, Y., Song, G., Wang, Y., Yang, X. , provided free of copyright via the Protein DataBank. View original data or read license terms.
