PDB | 8i7v Acipimox bound human hydroxy-carboxylic acid receptor 2

Cryo-EM structure of Acipimox bound human hydroxy-carboxylic acid receptor 2 in complex with Gi heterotrimer

label Keywords
gpcr, g-protein, membrane protein, acipimox, signaling
event_note Published
10/09/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
5-methyl-4-oxidanyl-pyrazin-4-ium-2-carboxylic acid

Original publication

import_contacts Title
Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.
import_contacts Journal
Nat Commun 2023
import_contacts DOI
10.1038/s41467-023-42764-8
person Authors
Ishimoto, N., Ohki, M., Kawakami, K., Tame, J.R.H., Lee, D.S., Ekimoto, T., Ikeguchi, M., Inoue, A., Park, S.Y., Park, J.H., Lee, Y.H., Ikuta, T.

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