PDB | 8i5g Structure of human Nav1.7

Structure of human Nav1.7 in complex with PF-05089771

label Keywords
inhibitor complex., membrane protein
event_note Published
10/23/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL HEMISUCCINATE, (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, PF-05089771, SODIUM ION, 1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE

Original publication

import_contacts Title
Structural mapping of Na v 1.7 antagonists.
import_contacts Journal
Nat Commun 2023
import_contacts DOI
10.1038/s41467-023-38942-3
person Authors
Wang, K., Pan, X., Huang, G., Huang, J., Jin, X., Wu, Q., Fan, X., Li, J., Yan, N.

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