PDB | 8i5b Structure of human Nav1.7

Structure of human Nav1.7 in complex with bupivacaine

label Keywords
inhibitor complex., membrane protein
event_note Published
10/16/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
2-acetamido-2-deoxy-beta-D-glucopyranose, O-[(R)-{[(2R)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine, CHOLESTEROL HEMISUCCINATE, 1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Levobupivacaine

Original publication

import_contacts Title
Structural mapping of Na v 1.7 antagonists.
import_contacts Journal
Nat Commun 2023
import_contacts DOI
10.1038/s41467-023-38942-3
person Authors
Wang, K., Pan, X., Huang, G., Huang, J., Jin, X., Wu, Q., Fan, X., Li, J., Yan, N.

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