PDB | 8i5b Structure of human Nav1.7
Structure of human Nav1.7 in complex with bupivacaine
label Keywords
inhibitor complex., membrane protein
event_note Published
10/16/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
2-acetamido-2-deoxy-beta-D-glucopyranose, O-[(R)-{[(2R)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine, CHOLESTEROL HEMISUCCINATE, 1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Levobupivacaine
Original publication
import_contacts Title
Structural mapping of Na v 1.7 antagonists.
import_contacts Journal
Nat Commun 2023
import_contacts DOI
10.1038/s41467-023-38942-3
person Authors
Wang, K., Pan, X., Huang, G., Huang, J., Jin, X., Wu, Q., Fan, X., Li, J., Yan, N.
Member of
copyrightData provided by Research Collaboration for Structural Biology, Wang, K., Pan, X., Huang, G., Huang, J., Jin, X., Wu, Q., Fan, X., Li, J., Yan, N. , provided free of copyright via the Protein DataBank. View original data or read license terms.