PDB | 8fsz Full-length mouse 5-HT3A receptor

Full-length mouse 5-HT3A receptor in complex with ALB148471, open-like

label Keywords
partial agonist, cys-loop, plgic, ion channel, transport protein
event_note Published
10/23/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
5-[(1R,3S,5R)-1-azabicyclo[3.2.2]nonan-3-yl]-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indazol-6-one, 2-acetamido-2-deoxy-beta-D-glucopyranose

Original publication

import_contacts Title
Structural basis for partial agonism in 5-HT 3A receptors.
import_contacts Journal
Nat.Struct.Mol.Biol. 2024
import_contacts DOI
10.1038/s41594-023-01140-2
person Authors
Felt, K., Huang, J., Filizola, M., Chakrapani, S., Salas-Estrada, L., Xie, D., Guzzo, P.R., Stauffer, M.

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