PDB | 8f6y Torpedo nicotinic acetylcholine receptor

Cryo-EM structure of Torpedo nicotinic acetylcholine receptor in complex with etomidate, desensitized-like state

label Keywords
acetylcholine receptor, nicotinic receptor, torpedo, cys-loop receptor, ion channel, muscle-type nicotinic receptor, transport protein-inhibitor complex, general anesthetic, inhibitor
event_note Published
11/13/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
Etomidate, CHOLINE ION, CHOLESTEROL, 2-acetamido-2-deoxy-beta-D-glucopyranose, (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, nonane

Original publication

import_contacts Title
Structural interplay of anesthetics and paralytics on muscle nicotinic receptors.
import_contacts Journal
Nat Commun 2023
import_contacts DOI
10.1038/s41467-023-38827-5
person Authors
Teng, J., Goswami, U., Hibbs, R.E., Rahman, M.M.

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