PDB | 7mby Human Cholecystokinin 1 receptor (CCK1R) Gq chimera (mGsqi) complex

Human Cholecystokinin 1 receptor (CCK1R) Gq chimera (mGsqi) complex

label Keywords
gpcr, membrane protein, membrane protein-signaling protein complex
event_note Published
11/06/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
CHOLESTEROL HEMISUCCINATE

Original publication

import_contacts Title
Structures of the human cholecystokinin 1 (CCK1) receptor bound to Gs and Gq mimetic proteins provide insight into mechanisms of G protein selectivity.
import_contacts Journal
Plos Biol. 2021
import_contacts DOI
10.1371/journal.pbio.3001295
person Authors
Sexton, P.M., Belousoff, M.J., Xu, X., Wootten, D., Venugopal, H., Miller, L.J., Harikumar, K.G., Danev, R., Mobbs, J.I., Thal, D.M., Christopoulos, A., Furness, S.G.B., Piper, S.J.

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