PDB | 6ur8 Human alpha4beta2 nicotinic acetylcholine receptor

CryoEM structure of human alpha4beta2 nicotinic acetylcholine receptor in complex with varenicline

label Keywords
acetylcholine receptor, nicotine, varenicline, membrane protein
event_note Published
11/13/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
2-acetamido-2-deoxy-beta-D-glucopyranose, VARENICLINE, beta-D-mannopyranose

Original publication

import_contacts Title
Synthetic antibodies against BRIL as universal fiducial marks for single-particle cryoEM structure determination of membrane proteins.
import_contacts Journal
Nat Commun 2020
import_contacts DOI
10.1038/s41467-020-15363-0
person Authors
Yeager, M., Coukos, J., Gao, X., Kang, Y., Radziwon, K., Skrobek, B.M., Purdy, M.D., Alvarez, F.J.D., Eric Xu, H., Dutka, P., Han, S., Ammirati, M., Kossiakoff, A.A., Fennell, K.F., Erramilli, S.K., Mukherjee, S., Qiu, X.

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