PDB | 6pbf ZINC9155420-bound TRPV5 in nanodiscs
ZINC9155420-bound TRPV5 in nanodiscs
label Keywords
trpv5, trp channel, inhibitor, calcium channel, transport protein
event_note Published
03/20/2024
filter_center_focus Method
ELECTRON MICROSCOPY
add_circle Ligands
(1S)-1-(4-oxo-5-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)ethyl [(2S)-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-2-yl]acetate
Original publication
import_contacts Title
Structure-based characterization of novel TRPV5 inhibitors.
import_contacts Journal
Elife 2019
import_contacts DOI
10.7554/eLife.49572
person Authors
Del Rosario, J.S., Yazici, A.T., Kapoor, A., Filizola, M., Rohacs, T., Fluck, E.C., Moiseenkova-Bell, V.Y., Hughes, T.E., Yudin, Y.
Member of
copyrightData provided by Research Collaboration for Structural Biology, Del Rosario, J.S., Yazici, A.T., Kapoor, A., Filizola, M., Rohacs, T., Fluck, E.C., Moiseenkova-Bell, V.Y., Hughes, T.E., Yudin, Y. , provided free of copyright via the Protein DataBank. View original data or read license terms.