PDB | 5x33 Leukotriene B4 receptor BLT1

Leukotriene B4 receptor BLT1 in complex with BIIL260

label Keywords
helix, membrane protein
event_note Published
11/20/2024
blur_on Resolution
3.7 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
4-[[3-[[4-[2-(4-hydroxyphenyl)propan-2-yl]phenoxy]methyl]phenyl]methoxy]benzenecarboximidamide

Original publication

import_contacts Title
Na+-mimicking ligands stabilize the inactive state of leukotriene B4receptor BLT1.
import_contacts Journal
Nat. Chem. Biol. 2018
import_contacts DOI
10.1038/nchembio.2547
person Authors
Yokomizo, T., Kawano, Y., Hirata, K., Yamamoto, M., Yamashita, K., Okuno, T., Hori, T., Hato, M., Shimizu, T., Yokoyama, S., Nakamura, M., Miyano, M.

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