PDB | 5l1h AMPA subtype ionotropic glutamate receptor GluA2

AMPA subtype ionotropic glutamate receptor GluA2 in complex with noncompetitive inhibitor GYKI53655

label Keywords
transporter, membrane protein, transport protein, transport protein-inhibitor complex
event_note Published
12/25/2024
blur_on Resolution
3.801 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
2-acetamido-2-deoxy-beta-D-glucopyranose, (8R)-5-(4-aminophenyl)-N,8-dimethyl-8,9-dihydro-2H,7H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-7-carboxamide

Original publication

import_contacts Title
Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
import_contacts Journal
Neuron 2016
import_contacts DOI
10.1016/j.neuron.2016.08.012
person Authors
Sampson, J.M., Yelshanskaya, M.V., Singh, A.K., Sobolevsky, A.I., Kurnikova, M., Narangoda, C.

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