PDB | 4zud Human Angiotensin Receptor
Crystal Structure of Human Angiotensin Receptor in Complex with Inverse Agonist Olmesartan at 2.8A resolution.
label Keywords
human angiotensin receptor at1r, bril, g protein-coupled receptor, gpcr, gpcr network, lipidic cubic phase, lcp, membrane protein, structural genomics, olmesartan, angiotensin receptor blocker, anti-hypertensive drug, psi-biology, signaling protein
event_note Published
11/06/2024
blur_on Resolution
2.8 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
Olmesartan
Original publication
import_contacts Title
Structural Basis for Ligand Recognition and Functional Selectivity at Angiotensin Receptor.
import_contacts Journal
J.Biol.Chem. 2015
import_contacts DOI
10.1074/jbc.M115.689000
person Authors
Karnik, S.S., Patel, N., Unal, H., Cherezov, V., Han, G.W., Katritch, V., Zhang, H., Desnoyer, R., Stevens, R.C.
Member of
copyrightData provided by Research Collaboration for Structural Biology, Karnik, S.S., Patel, N., Unal, H., Cherezov, V., Han, G.W., Katritch, V., Zhang, H., Desnoyer, R., Stevens, R.C. , provided free of copyright via the Protein DataBank. View original data or read license terms.