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      PDB | 3zpr Thermostabilised turkey beta1 adrenergic receptor

      Thermostabilised turkey beta1 adrenergic receptor with 4-methyl-2-(piperazin-1-yl) quinoline bound

      label Keywords
      membrane protein, gpcr, fragment screening, aryl piperazine, structure based drug design
      event_note Published
      10/23/2024
      blur_on Resolution
      2.7 Å
      filter_center_focus Method
      X-RAY DIFFRACTION
      add_circle Ligands
      SODIUM ION, CHOLESTEROL HEMISUCCINATE, 4-METHYL-2-(PIPERAZIN-1-YL) QUINOLINE, HEGA-10

      Original publication

      import_contacts Title
      Biophysical Fragment Screening of the Beta1-Adrenergic Receptor: Identification of High Affinity Aryl Piperazine Leads Using Structure-Based Drug Design.
      import_contacts Journal
      J.Med.Chem. 2013
      import_contacts DOI
      10.1021/JM400140Q
      person Authors
      Warne, T., Errey, J., Congreve, M., Marshall, F.H., Tehan, B., Dore, A., Christopher, J., Brown, J., Tate, C.G., Koglin, M., Rich, R.L., Myszka, D.

      Read article from J.Med.Chem.

      copyrightData provided by Research Collaboration for Structural Biology, Warne, T., Errey, J., Congreve, M., Marshall, F.H., Tehan, B., Dore, A., Christopher, J., Brown, J., Tate, C.G., Koglin, M., Rich, R.L., Myszka, D. , provided free of copyright via the Protein DataBank. View original data or read license terms.

      Simulations available

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