PDB | 3w9h Structural basis for the inhibition of bacterial multidrug exporters
Structural basis for the inhibition of bacterial multidrug exporters
label Keywords
acrb, efflux pump, transporter, multidrug efflux pump, acra, tolc, inner membrane, transport protein, membrane protein
event_note Published
04/04/2013
blur_on Resolution
3.05 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
[{2-[({[(3R)-1-{8-[(4-tert-butyl-1,3-thiazol-2-yl)carbamoyl]-4-oxo-3-[(E)-2-(1H-tetrazol-5-yl)ethenyl]-4H-pyrido[1,2-a]pyrimidin-2-yl}piperidin-3-yl]oxy}carbonyl)amino]ethyl}(dimethyl)ammonio]acetate
Original publication
import_contacts Title
Structural basis for the inhibition of bacterial multidrug exporters
import_contacts Journal
Nature 2013
import_contacts DOI
10.1038/nature12300
person Authors
Sakurai, K., Yamaguchi, A., Nagata, C., Nishino, K., Yamasaki, S., Hayashi, K., Hoshino, K., Nakashima, R., Onodera, Y.
copyrightData provided by Research Collaboration for Structural Biology, Sakurai, K., Yamaguchi, A., Nagata, C., Nishino, K., Yamasaki, S., Hayashi, K., Hoshino, K., Nakashima, R., Onodera, Y. , provided free of copyright via the Protein DataBank. View original data or read license terms.