PDB | 3w9h Structural basis for the inhibition of bacterial multidrug exporters

Structural basis for the inhibition of bacterial multidrug exporters

label Keywords
acrb, efflux pump, transporter, multidrug efflux pump, acra, tolc, inner membrane, transport protein, membrane protein
event_note Published
04/04/2013
blur_on Resolution
3.05 Å
filter_center_focus Method
X-RAY DIFFRACTION
add_circle Ligands
[{2-[({[(3R)-1-{8-[(4-tert-butyl-1,3-thiazol-2-yl)carbamoyl]-4-oxo-3-[(E)-2-(1H-tetrazol-5-yl)ethenyl]-4H-pyrido[1,2-a]pyrimidin-2-yl}piperidin-3-yl]oxy}carbonyl)amino]ethyl}(dimethyl)ammonio]acetate

Original publication

import_contacts Title
Structural basis for the inhibition of bacterial multidrug exporters
import_contacts Journal
Nature 2013
import_contacts DOI
10.1038/nature12300
person Authors
Sakurai, K., Yamaguchi, A., Nagata, C., Nishino, K., Yamasaki, S., Hayashi, K., Hoshino, K., Nakashima, R., Onodera, Y.

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